FL-CARES Cancer Data
Resources
Cancer Drugs
Compounds
Diseases
Targets
Data Sources
Identifiers
About this Project
Taletrectinib
US FDA Label
Compound
: 3-[4-[(2R)-2-aminopropoxy]phenyl]-N-[(1R)-1-(3-fluorophenyl)ethyl]imidazo[1,2-b]pyridazin-6-amine
Description:
Taletrectinib is an orally available small molecule kinase inhibitor. It is targeted against ROS1, including resistant mutant forms, and shows some inhibitor activity against tropomyosin receptor kinases (TRKs) TRKA, TRKB, and TRKC.
Brand Name:
Code(s):
AB106
Approved:
Kinase Class:
RY
Inhibitor Type:
?
Literature (PubMed):
0
Target(s):
epidermal growth factor receptor
Disease(s):
non-small-cell lung carcinoma
Identifiers (4)
International Nonproprietary Name
: Taletrectinib [INN] (Source: PubChem)
KEGG Drug ID
: D12363 (Source: PubChem)
USFDA Precision ID
: UNII-W4141180YD (Source: PubChem)
US Adopted Name
: Taletrectinib [USAN] (Source: PubChem)